SCHEMBL28229042

SCHEMBL28229042

O=C(O)c1ccc2c(c1)CCN2.O=C(O)c1ccc2c(c1)NCC2

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.71
MAPT P10636 3/20 0.71
ALDH1A1 P00352 3/20 0.50
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44
ACHE P22303 3/20 0.43
CRBN Q96SW2 2/20 0.43
SRD5A2 P31213 4/20 0.41
SRD5A1 P18405 3/20 0.41
GFER P55789 1/20 0.41
POLB P06746 1/20 0.41
BLM P54132 1/20 0.41
GRM1 Q13255 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2638095 0.93 KDM4E (0.81) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL3096217 0.93 KDM4E (0.60) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL29906797 0.93 KDM4E (0.60) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL29530477 0.93 KDM4E (0.81) KDM4EMAPTALDH1A1DRD2DRD4
Hydrochloric Acid SCHEMBL698487 0.92 KDM4E (0.78) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL45202 0.83 KDM4E (1.00) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL29365830 0.83 KDM4E (0.76) KDM4EMAPTALDH1A1ACHESRD5A2
SCHEMBL2730135 0.83 KDM4E (0.76) KDM4EMAPTALDH1A1ACHESRD5A2
SCHEMBL29673258 0.83 KDM4E (1.00) KDM4EMAPTALDH1A1DRD2DRD4
SCHEMBL4051485 0.81 KDM4E (0.58) KDM4EMAPTALDH1A1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108276382-A Cell cycle protein dependent kinase inhibitor and its application 南京圣和药业股份有限公司 2018-07-13 CN disclosed