SCHEMBL28229249

SCHEMBL28229249

Cc1cccc(NCc2ccccc2)c1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.53
HSD17B10 Q99714 2/20 0.50
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CRHBP P24387 1/20 0.44
CYP2C19 P33261 1/20 0.44
CRHR2 Q13324 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3440796 0.83 ADRA2C (0.72) ADRA2CHSD17B10HDAC1HDAC8HDAC6
SCHEMBL2232108 0.81 HSD17B10 (0.60) ADRA2CHSD17B10KDM4EHPGDTSHR
Bromide SCHEMBL30496129 0.81 ADRA2C (0.70) ADRA2CHSD17B10HDAC1HDAC8HDAC6
Bromide SCHEMBL29049211 0.80 HSD17B10 (0.58) ADRA2CHSD17B10KDM4EHPGDTSHR
Ammonia Solution, Strong SCHEMBL28850909 0.80 HSD17B10 (0.58) ADRA2CHSD17B10KDM4EHPGDTSHR
Hydrochloric Acid SCHEMBL4373569 0.80 HSD17B10 (0.58) ADRA2CHSD17B10KDM4EHPGDTSHR
Iodide SCHEMBL29049215 0.80 HSD17B10 (0.58) ADRA2CHSD17B10KDM4EHPGDTSHR
Water SCHEMBL29049225 0.80 HSD17B10 (0.58) ADRA2CHSD17B10KDM4EHPGDTSHR
SCHEMBL5608826 0.79 HTT (0.53) ADRA2CKDM4EHPGDTSHRHTT
SCHEMBL12956811 0.79 HTT (0.46) ADRA2CHDAC1HDAC8HDAC6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105859651-B Thiazole derivative and its synthetic method and application 华东师范大学 2018-06-22 CN disclosed