SCHEMBL2823209

SCHEMBL2823209

COc1cc(C=CC(=O)NCc2cccc(CCc3ccccc3)c2)ccc1-n1ccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
KDM4E B2RXH2 6/20 0.51
HPGD P15428 3/20 0.49
POLB P06746 2/20 0.49
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
MAPT P10636 2/20 0.48
ALOX5 P09917 1/20 0.48
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
MMP1 P03956 2/20 0.45
MMP2 P08253 2/20 0.45
MMP9 P14780 2/20 0.45
APP P05067 1/20 0.45
THRB P10828 1/20 0.45
LMNA P02545 2/20 0.44
PRNP P04156 1/20 0.44
GAA P10253 1/20 0.44
BLM P54132 1/20 0.44
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823206 1.00 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDPOLBMAOA
Trifluoroacetic Acid SCHEMBL1238716 0.95 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDPOLBMAOA
Trifluoroacetic Acid SCHEMBL1238713 0.95 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDPOLBMAOA
SCHEMBL14870573 0.93 KDM4E (0.55) ALDH1A1KDM4EHPGDPOLBMAOA
SCHEMBL14870574 0.89 KDM4E (0.50) ALDH1A1KDM4EHPGDPOLBMAPT
SCHEMBL1239255 0.89 KDM4E (0.50) ALDH1A1KDM4EHPGDPOLBMAPT
SCHEMBL1239258 0.89 KDM4E (0.50) ALDH1A1KDM4EHPGDPOLBMAPT
SCHEMBL12712438 0.86 KDM4E (0.48) ALDH1A1KDM4EHPGDPOLBMAOA
SCHEMBL14870580 0.85 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDPOLBMAPT
SCHEMBL1239838 0.84 KDM4E (0.48) ALDH1A1KDM4EHPGDPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2261218-A2 Process for preparing phenyl-, pyridinyl- or pyrimidinyl-substituted imidazoles Eisai R&D Management Co., Ltd. (JP) 2010-12-15 EP disclosed