SCHEMBL28236753

SCHEMBL28236753

CNc1ccc(-n2cccn2)nc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.54
ALDH1A1 P00352 3/20 0.54
RXFP1 Q9HBX9 1/20 0.54
LMNA P02545 1/20 0.53
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
HPGD P15428 2/20 0.48
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2D6 P10635 1/20 0.47
CXCR4 P61073 1/20 0.43
NAMPT P43490 1/20 0.42
CHRNA7 P36544 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TNIK Q9UKE5 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24922507 0.77 ADORA2A (0.46) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL46317 0.77 KDM4E (0.58) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL31516755 0.77 KDM4E (0.58) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL3462062 0.77 LMNA (0.57) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL10754057 0.77 CXCR4 (0.53) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL19796113 0.76 NAMPT (0.50) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL11117073 0.75 NOTUM (0.58) KDM4EALDH1A1RXFP1KMT2AMEN1
SCHEMBL23957682 0.75 LMNA (0.48) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL2728318 0.74 LMNA (0.57) KDM4EALDH1A1RXFP1LMNAKMT2A
SCHEMBL22925970 0.74 LMNA (0.57) KDM4EALDH1A1RXFP1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881683-A PI3K alpha inhibitors and methods of use thereof 传达治疗有限公司 2024-04-12 CN disclosed
CN-116730978-A Compound containing heteroaromatic ring alkynyl, preparation method and application thereof 中国科学院上海药物研究所 2023-09-12 CN disclosed
CN-114702495-A Purinones as ubiquitin-specific protease 1 inhibitors 福马治疗有限公司 2022-07-05 CN disclosed
CN-108473495-B Purinones as ubiquitin-specific protease 1 inhibitors 福马治疗有限公司 2022-04-12 CN disclosed
CN-108473495-A Purinones as ubiquitin-specific protease 1 inhibitors 福马治疗有限公司 2018-08-31 CN disclosed