SCHEMBL2823746

SCHEMBL2823746

CC(Cc1ccc(OCC(F)(F)c2ccccc2)cc1)NC[C@@H](O)c1ccc(O)c(NC=O)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 12/20 0.69
ADRB1 P08588 6/20 0.69
ADRB3 P13945 5/20 0.69
DRD2 P14416 2/20 0.69
CYP1A2 P05177 2/20 0.69
CYP3A4 P08684 2/20 0.69
CYP2D6 P10635 2/20 0.69
TSHR P16473 2/20 0.69
MAPK1 P28482 2/20 0.69
PGR P06401 1/20 0.69
SLC6A4 P31645 1/20 0.69
ADRA1A P35348 1/20 0.69
PTGS2 P35354 1/20 0.69
SLC6A3 Q01959 1/20 0.69
CYP2C19 P33261 1/20 0.69
DRD3 P35462 1/20 0.69
NFKB1 P19838 1/20 0.51
RAB9A P51151 1/20 0.51
HIF1A Q16665 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823742 1.00 ADRB2 (0.69) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL2823750 1.00 ADRB2 (0.69) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL13232144 1.00 ADRB2 (0.69) ADRB2ADRB1ADRB3DRD2CYP1A2
Formic Acid SCHEMBL2792055 0.98 ADRB2 (0.67) ADRB2ADRB1ADRB3DRD2CYP1A2
Formic Acid SCHEMBL2792049 0.98 ADRB2 (0.67) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL2793400 0.89 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL2793403 0.89 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL2853299 0.85 ADRB2 (0.54) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL2853304 0.85 ADRB2 (0.54) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL13232147 0.85 ADRB2 (0.74) ADRB2ADRB1ADRB3DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057122-B1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE 2 ADRENERGIC RECEPTOR ALMIRALL SA (ES) 2010-09-01 EP claimed
EP-2057122-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE 2 ADRENERGIC RECEPTOR Laboratorios Almirall, S.A. (ES) 2009-05-13 EP claimed
WO-2008046598-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE β2 ADRENERGIC RECEPTOR LABORATORIOS ALMIRALL, S.A. (ES) 2008-04-24 WO claimed
EP-2057122-B1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE 2 ADRENERGIC RECEPTOR ALMIRALL SA (ES) 2010-09-01 EP disclosed