SCHEMBL28237663

SCHEMBL28237663

COCCn1cc2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.46
HPGD P15428 3/20 0.44
IRAK4 Q9NWZ3 2/20 0.41
KDM4E B2RXH2 5/20 0.40
RAB9A P51151 4/20 0.40
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
GLA P06280 3/20 0.40
GAA P10253 3/20 0.40
NPC1 O15118 3/20 0.40
TSHR P16473 4/20 0.39
CASR P41180 1/20 0.39
LMNA P02545 3/20 0.38
HSD17B10 Q99714 2/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 1/20 0.38
RECQL P46063 1/20 0.38
AR P10275 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30177201 0.90 IRAK4 (0.43) MPOHPGDIRAK4KDM4ERAB9A
SCHEMBL10123647 0.80 SLC6A2 (0.44) HPGDKDM4ERAB9AALDH1A1SMN1; SMN2
SCHEMBL13607537 0.80 IRAK4 (0.39) MPOHPGDIRAK4KDM4ERAB9A
SCHEMBL30995500 0.79 MAP4K4 (0.43) IRAK4KDM4ERAB9AALDH1A1TSHR
SCHEMBL14909598 0.79 KDM4E (0.58) MPOHPGDIRAK4KDM4ERAB9A
SCHEMBL25219391 0.79 NFATC1 (0.42) MPOIRAK4ALDH1A1HSD17B10
SCHEMBL28505047 0.79 IRAK4 (0.32) IRAK4KDM4EALDH1A1GAAKMT2A
SCHEMBL13607538 0.79 IRAK4 (0.41) HPGDIRAK4KDM4ERAB9AALDH1A1
SCHEMBL19128033 0.78 IRAK4 (0.36) MPOHPGDIRAK4KDM4EALDH1A1
SCHEMBL24338409 0.78 IRAK4 (0.43) MPOIRAK4KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108473471-A Substituted thiourocystine derivatives as androgen receptor antagonists 詹森药业有限公司 2018-08-31 CN claimed
CN-108473471-A Substituted thiourocystine derivatives as androgen receptor antagonists 詹森药业有限公司 2018-08-31 CN disclosed