SCHEMBL28237753

SCHEMBL28237753

O=C(c1ccc(-n2cc(-c3ccc4ccc(=O)[nH]c4c3)nn2)cc1)N1CCOCC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.46
RIPK1 Q13546 1/20 0.43
LRRK2 Q5S007 1/20 0.43
HPGD P15428 5/20 0.43
JAK2 O60674 1/20 0.42
MGLL Q99685 6/20 0.42
STIM1 Q13586 1/20 0.41
ORAI1 Q96D31 1/20 0.41
HTR2B P41595 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GPR84 Q9NQS5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28238879 0.84 HPGD (0.51) RIPK1HPGDMGLL
SCHEMBL19146343 0.81 PIK3CA (0.45) PIK3CARIPK1LRRK2HPGDJAK2
SCHEMBL19126423 0.81 PIK3CA (0.45) PIK3CALRRK2HPGDALDH1A1
SCHEMBL19126328 0.81 PIK3CA (0.45) PIK3CALRRK2MGLLHTR2BALDH1A1
SCHEMBL19126428 0.81 PIK3CA (0.45) PIK3CALRRK2HPGDHTR2B
SCHEMBL19126514 0.81 PIK3CA (0.45) PIK3CAHPGDJAK2ALDH1A1
SCHEMBL28238897 0.81 HPGD (0.48) HPGDMGLLALDH1A1
SCHEMBL19126670 0.81 ALK (0.46) PIK3CALRRK2HTR2B
SCHEMBL19144550 0.80 POLB (0.50) PIK3CARIPK1HPGDMGLLHTR2B
SCHEMBL19127065 0.79 ALDH1A1 (0.46) PIK3CAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108473485-A QUINOLIN-2-ONE DERIVATIVES 默克专利股份公司 2018-08-31 CN claimed
CN-108473485-A QUINOLIN-2-ONE DERIVATIVES 默克专利股份公司 2018-08-31 CN disclosed