SCHEMBL28239121

SCHEMBL28239121

CC1(C)c2ccccc2C=CC1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
DRD2 P14416 1/20 0.31
CHRM3 P20309 1/20 0.31
DRD1 P21728 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
ADRA1A P35348 1/20 0.31
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK4 Q16654 1/20 0.31
CACNB4 O00305 1/20 0.31
CACNA1A O00555 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNG3 O60359 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18394586 0.78 KDM4E (0.32) KDM4EPKMPDK2PDK4
SCHEMBL28239549 0.76 KDM4E (0.31) KDM4EPKMPDK2PDK4
SCHEMBL28240050 0.76 KDM4E (0.31) KDM4EPKMPDK2PDK4
SCHEMBL15716844 0.76 PDK2 (0.34) KDM4EPKMPDK2PDK4
SCHEMBL7610207 0.76 HTR2A (0.32) KDM4EPKMHTR2APDK2PDK4
SCHEMBL15717305 0.74 PDK2 (0.33) KDM4EPKMPDK2PDK4
SCHEMBL6537805 0.73 KDM4E (0.36) KDM4EPKM
SCHEMBL28021929 0.73 KDM4E (0.40) KDM4EPKM
SCHEMBL7649583 0.71 KDM4E (0.31) KDM4EPKM
SCHEMBL28228066 0.69 THRB (0.38) KDM4EPKMCACNB4CACNA1ACACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903310-B Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain 阵列生物制药公司 2018-08-14 CN disclosed