SCHEMBL28241995

SCHEMBL28241995

N#Cc1ccccc1CON=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
HTT P42858 1/20 0.46
MEN1 O00255 1/20 0.46
FFAR1 O14842 1/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 1/20 0.43
TSHR P16473 1/20 0.42
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
PLAU P00749 1/20 0.40
ALKBH1 Q13686 1/20 0.40
MAOB P27338 1/20 0.40
CYP19A1 P11511 1/20 0.39
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17986342 0.83 RAB9A (0.47) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17217989 0.79 RAB9A (0.44) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17986285 0.79 RAB9A (0.50) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17986286 0.79 RAB9A (0.50) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17217987 0.79 RAB9A (0.44) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL6668462 0.78 FFAR1 (0.46) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL28106820 0.77 RAB9A (0.55) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17218254 0.77 RAB9A (0.43) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17218250 0.77 RAB9A (0.43) RAB9AKMT2ANPC1TDP1HTT
SCHEMBL17218959 0.76 RAB9A (0.45) RAB9AKMT2ANPC1TDP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110066273-A A kind of single arylpyrimidines HIV-1 reverse transcriptase inhibitor of the ring containing triazole and the preparation method and application thereof 山东大学 2019-07-30 CN claimed
CN-109705095-A A kind of condensed ring 1,4-benzoquinone class CDC25 protein phosphatase inhibitor of the ring containing triazole and its preparation method and application 山东大学 2019-05-03 CN claimed
CN-108586482-A A kind of Diarylmiazines HIV-1 inhibitor of the ring containing triazole and its preparation method and application 山东大学 2018-09-28 CN claimed
CN-108586482-A A kind of Diarylmiazines HIV-1 inhibitor of the ring containing triazole and its preparation method and application 山东大学 2018-09-28 CN disclosed