Quinoline

Quinoline

SCHEMBL28245218

O=[N+]([O-])c1ccnc2ccccc12.c1ccc2ncccc2c1

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.73
NCOA1 Q15788 1/20 0.59
NCOA3 Q9Y6Q9 1/20 0.59
CYP1A2 P05177 1/20 0.54
TSHR P16473 1/20 0.54
ALDH1A1 P00352 10/20 0.53
MAPT P10636 7/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
PDE10A Q9Y233 1/20 0.49
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
KDM4E B2RXH2 5/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
LMNA P02545 4/20 0.48
TDP1 Q9NUW8 4/20 0.48
HTT P42858 3/20 0.48
CTSB P07858 2/20 0.48
IDO1 P14902 2/20 0.48
TDO2 P48775 2/20 0.48
HSP90AA1 P07900 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL9110913 0.94 POLB (0.84) POLBNCOA1NCOA3CYP1A2TSHR
SCHEMBL538895 0.90 POLB (0.77) POLBNCOA1NCOA3CYP1A2TSHR
SCHEMBL30531716 0.89 POLB (0.74) POLBNCOA1NCOA3CYP1A2TSHR
SCHEMBL29611471 0.85 POLB (1.00) POLBNCOA1NCOA3CYP1A2TSHR
SCHEMBL827685 0.85 POLB (1.00) POLBNCOA1NCOA3CYP1A2TSHR
SCHEMBL29750649 0.85 POLB (1.00) POLBNCOA1NCOA3CYP1A2TSHR
Quinoline SCHEMBL27814435 0.85 POLB (0.64) POLBNCOA1NCOA3CYP1A2TSHR
Hydrochloric Acid SCHEMBL7950313 0.83 POLB (0.96) POLBNCOA1NCOA3CYP1A2TSHR
Quinoline SCHEMBL28344417 0.80 ALDH1A1 (0.52) POLBNCOA1NCOA3CYP1A2TSHR
Quinoline SCHEMBL28125435 0.80 POLB (0.61) POLBNCOA1NCOA3CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108610286-A A kind of 2- aryl-4-quinolones derivative and its preparation method and application 绍兴文理学院 2018-10-02 CN disclosed