SCHEMBL28245455

SCHEMBL28245455

O=C(O)c1cc(Cn2ncc3ccccc3c2=O)ccc1F

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.60
RXFP1 Q9HBX9 3/20 0.46
PKM P14618 3/20 0.46
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MITF O75030 1/20 0.44
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
PLA2G10 O15496 1/20 0.43
POLB P06746 3/20 0.42
GAA P10253 2/20 0.41
APOBEC3G Q9HC16 1/20 0.41
PTGER4 P35408 1/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31140178 0.82 PARP1 (0.57) TDP1
SCHEMBL30495895 0.82 TDP1 (0.50) TDP1
SCHEMBL31656091 0.81 PARP1 (0.59) TDP1
Hydrochloric Acid SCHEMBL2253051 0.81 PTGER4 (0.41) TDP1ALDH1A1KDM4ELMNAGAA
SCHEMBL28244751 0.80 TDP1 (0.60) TDP1PKMALDH1A1NPC1RAB9A
SCHEMBL29703239 0.79 TDP1 (0.69) TDP1RXFP1PKMALDH1A1NPC1
SCHEMBL7894526 0.79 TDP1 (0.69) TDP1RXFP1PKMALDH1A1NPC1
SCHEMBL29463417 0.78 PARP1 (0.56) TDP1
SCHEMBL30141798 0.78 PARP1 (0.48) TDP1
SCHEMBL29703247 0.78 TDP1 (0.72) TDP1RXFP1PKMALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558773-A A kind of preparation method of olaparib pharmaceutical intermediate 苏州莱克施德药业有限公司 2018-09-21 CN disclosed