SCHEMBL2824740

SCHEMBL2824740

NS(=O)(=O)c1ccc(C#Cc2cnn3ccc(-c4ccc(Cl)cc4)cc23)s1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.32
CA2 P00918 4/20 0.32
CA9 Q16790 4/20 0.32
CA1 P00915 3/20 0.32
EPHB3 P54753 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
SCN5A Q14524 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1348859 0.81 SMN1; SMN2 (0.39) CA12CA2CA9CA1PTGS1
SCHEMBL1348308 0.73 HPGD (0.35) CA12CA2CA9CA1PTGS1
SCHEMBL1350177 0.71 HPGD (0.43)
SCHEMBL1348844 0.71 CSNK2A1 (0.32) CA12CA2CA9CA1PTGS2
SCHEMBL1348845 0.71 HPGD (0.35) CA12CA2CA9CA1PTGS1
SCHEMBL1349028 0.71 PSD (0.34) CA12CA2CA9CA1
SCHEMBL1348457 0.69 HPGD (0.36) CA2CA9CA1PTGS1PTGS2
SCHEMBL1348119 0.69 CA12 (0.38) CA12CA2CA9CA1PTGS2
SCHEMBL2854594 0.69 KDM4E (0.34) SCN5A
SCHEMBL1348046 0.67 CA12 (0.32) CA12CA2CA9CA1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863818-B1 ACETYLENYL-PYRAZOLO-PVRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-03-10 EP disclosed