SCHEMBL2854594

SCHEMBL2854594

NS(=O)(=O)c1ccc(C#Cc2cnn3ccc(-c4ccc(C(F)F)cc4)nc23)s1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SCN5A Q14524 2/20 0.32
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1348859 0.87 SMN1; SMN2 (0.39) KDM4EALDH1A1SMN1; SMN2L3MBTL1SCN5A
SCHEMBL1348729 0.75 LMNA (0.38) KDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1348596 0.71 POLB (0.38) KDM4EALDH1A1SMN1; SMN2
SCHEMBL1348807 0.70 HPGD (0.43) KDM4EALDH1A1L3MBTL1
SCHEMBL1348308 0.70 HPGD (0.35) KDM4EALDH1A1SMN1; SMN2
SCHEMBL1350177 0.70 HPGD (0.43) KDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1348486 0.70 CA12 (0.37) KDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1348507 0.69 LMNA (0.38) KDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1346184 0.69 TTR (0.40) KDM4EALDH1A1L3MBTL1
SCHEMBL1348845 0.68 HPGD (0.35) KDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863818-B1 ACETYLENYL-PYRAZOLO-PVRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-03-10 EP disclosed