SCHEMBL2825003

SCHEMBL2825003

CCOC(=O)c1cc(Br)cc(C#N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.50
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
CA7 P43166 3/20 0.50
CA9 Q16790 3/20 0.50
CA14 Q9ULX7 3/20 0.50
GPR35 Q9HC97 1/20 0.43
ESR1 P03372 3/20 0.42
ESR2 Q92731 1/20 0.42
KDM4E B2RXH2 4/20 0.41
GLA P06280 1/20 0.41
ATM Q13315 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747236 0.84 CYP2C9 (0.55) CA12CA1CA2CA7CA9
SCHEMBL5224940 0.83 NOTUM (0.53) CA12CA1CA2CA7CA9
SCHEMBL8446374 0.83 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL31237155 0.83 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL23384739 0.83 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL2712707 0.82 CA12 (0.64) CA12CA1CA2CA7CA9
SCHEMBL10180584 0.82 CA12 (0.64) CA12CA1CA2CA7CA9
SCHEMBL5102877 0.79 GABRA1 (0.39) CA12CA1CA2CA9CA14
SCHEMBL4693441 0.79 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL9743746 0.78 CA12 (0.55) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069504-A1 (3-OXO)PYRIDIN-4-YLUREA DERIVATIVES AS PDE4 INHIBITORS ALMIRALL, S.A. (ES) 2010-06-24 WO disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed