SCHEMBL28256351

SCHEMBL28256351

Cc1c[nH]nc1NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.39
CA1 P00915 2/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
CYP17A1 P05093 1/20 0.37
ATR Q13535 1/20 0.37
GFER P55789 2/20 0.36
BRD9 Q9H8M2 1/20 0.36
BRD4 O60885 1/20 0.36
CA2 P00918 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955035 0.81 CYP17A1 (0.38) LCKCA1CA12CA9CYP17A1
SCHEMBL7432621 0.81 ATR (0.41) CA1KDM4ELMNACYP17A1ATR
SCHEMBL16770460 0.81 ATR (0.38) CA1KDM4ELMNACYP17A1ATR
SCHEMBL19026780 0.80 RAB9A (0.36) CA1CYP17A1ATRCA2
SCHEMBL18138246 0.78 PRMT1 (0.41) LMNACYP17A1ATRALDH1A1
SCHEMBL27164185 0.78 CYP17A1 (0.36) CA1KDM4ELMNACYP17A1ATR
SCHEMBL4015102 0.77 BRD9 (0.39) LCKCA1CYP17A1ATRBRD9
SCHEMBL20555276 0.74 GSK3B (0.39) LCKCA1CA12CA9CYP17A1
SCHEMBL15264820 0.73 ATR (0.48) CA1CYP17A1ATRCA2
SCHEMBL22621090 0.72 LCK (0.46) LCKCA1CA12CA9CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884050-A Tetrahydroisoquinoline derivatives UCB生物制药私人有限公司 2018-11-23 CN disclosed