SCHEMBL28258100

SCHEMBL28258100

FC(F)(F)Cn1ccc2c(I)cccc21

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ASH1L Q9NR48 2/20 0.41
HTR2C P28335 4/20 0.36
HTR2A P28223 2/20 0.36
NR3C1 P04150 3/20 0.33
PGR P06401 3/20 0.33
NR3C2 P08235 3/20 0.33
HTR6 P50406 2/20 0.33
CYP17A1 P05093 3/20 0.32
CYP1A2 P05177 1/20 0.32
HTR3A P46098 2/20 0.32
CCR4 P51679 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12825335 0.80 CCR4 (0.41) HTR2CHTR2AHTR6CCR4
SCHEMBL14981465 0.79 HTR2C (0.55) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL14977330 0.79 ASH1L (0.41) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL29811286 0.79 ASH1L (0.41) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL30595498 0.79 ASH1L (0.39) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL30098925 0.76 IDO1 (0.44) ASH1LHTR6HTR3A
SCHEMBL30098893 0.76 HTR6 (0.42) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL28826241 0.76 HTR6 (0.60) ASH1LHTR2CHTR2ANR3C1PGR
SCHEMBL19260954 0.74 KDM4E (0.43) ASH1LNR3C1PGRNR3C2CYP1A2
SCHEMBL30098951 0.74 HTR2C (0.36) ASH1LHTR2CHTR2ANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109069481-A Methods and compounds for restoring function of mutant p53 皮姆维制药公司 2018-12-21 CN disclosed