SCHEMBL28259104

SCHEMBL28259104

FC(F)(F)c1ccnc2ccc(Cl)cc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.56
CDK8 P49336 2/20 0.44
DAPK3 O43293 1/20 0.44
ABL1 P00519 1/20 0.44
PDGFRB P09619 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
ACVR1 Q04771 1/20 0.44
TYRO3 Q06418 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
AAK1 Q2M2I8 1/20 0.44
SOS2 Q07890 1/20 0.43
SLC40A1 Q9NP59 1/20 0.43
AR P10275 2/20 0.42
CCNC P24863 1/20 0.41
CNR1 P21554 1/20 0.41
PARP1 P09874 1/20 0.41
GAK O14976 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669631 0.86 NR4A2 (0.56) NR4A2ABL1GSK3AGSK3BACVR1
SCHEMBL28029894 0.83 AR (0.49) NR4A2ARCNR1CYP1A2MAPT
SCHEMBL11891560 0.82 NR4A2 (0.56) NR4A2CDK8PDGFRBAAK1SOS2
SCHEMBL30632276 0.80 CDK8 (0.46) CDK8CLK2ACVR1CLK4DYRK1B
SCHEMBL20392593 0.79 SLC22A12 (0.52) CDK8ABL1ACVR1AAK1AR
SCHEMBL28819002 0.79 RIPK2 (0.47) ARPARP1RIPK2MAPTKMT2A
SCHEMBL3935913 0.79 HTR1A (0.50) CDK8ACVR1CLK4ARPARP1
SCHEMBL13676600 0.76 RIPK2 (0.45) CDK8ABL1CLK2GSK3BCLK4
SCHEMBL10914959 0.75 AR (0.44) ARHCAR1MAPTSMN1; SMN2
SCHEMBL30051309 0.75 NR4A2 (0.66) NR4A2CDK8DYRK1BSOS2CCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884061-A 1,2,4- triazine -3- amine derivant, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-11-23 CN disclosed