SCHEMBL28260795

SCHEMBL28260795

CC(Br)c1ncnc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.47
PI4K2B Q8TCG2 1/20 0.47
PI4K2A Q9BTU6 1/20 0.47
PI4KB Q9UBF8 1/20 0.47
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
GALR3 O60755 1/20 0.46
NR2F2 P24468 1/20 0.46
ADORA2A P29274 2/20 0.44
EGFR P00533 2/20 0.42
BCAT2 O15382 1/20 0.42
DAPK3 O43293 1/20 0.41
MAP4K4 O95819 1/20 0.41
ABL1 P00519 1/20 0.41
ERBB2 P04626 1/20 0.41
PIM1 P11309 1/20 0.41
PRKACA P17612 1/20 0.41
LTK P29376 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6371765 0.86 PI4KA (0.52) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL20115779 0.78 PI4KA (0.44) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL21362866 0.75 SMN1; SMN2 (0.43) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL30838566 0.71 LMNA (0.44) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL7486261 0.70 PI4KA (0.48) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL10562950 0.70 MAPT (0.48) NPC1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL3951708 0.69 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL637552 0.69 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL22918311 0.68 SMN1; SMN2 (0.54) PI4KAPI4K2BPI4K2API4KBPDE4A
SCHEMBL803121 0.68 PI4KA (0.50) PI4KAPI4K2BPI4K2API4KBPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884061-A 1,2,4- triazine -3- amine derivant, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-11-23 CN disclosed