SCHEMBL28274262

SCHEMBL28274262

N#Cc1c[nH]c2nc(Cl)ncc12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 7/20 0.47
CSNK1A1 P48729 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
CHUK O15111 2/20 0.44
DYRK1A Q13627 2/20 0.40
PIN1 Q13526 1/20 0.39
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
HASPIN Q8TF76 1/20 0.38
RPS6KA5 O75582 2/20 0.37
IMPDH2 P12268 1/20 0.37
IMPDH1 P20839 1/20 0.37
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
CDC42BPA Q5VT25 2/20 0.36
CDC42BPB Q9Y5S2 2/20 0.36
TYRO3 Q06418 1/20 0.35
DYRK1B Q9Y463 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30899087 1.00 LRRK2 (0.47) LRRK2CSNK1A1CLK4CHUKDYRK1A
SCHEMBL31586107 0.79 LRRK2 (0.47) LRRK2CHUKCCNT1CDK9HASPIN
SCHEMBL25401085 0.79 CHUK (0.51) LRRK2CHUK
SCHEMBL22518633 0.76 RPS6KA5 (0.45) LRRK2RPS6KA5TYRO3DYRK1B
SCHEMBL26638109 0.76 LRRK2 (0.44) LRRK2CHUKCCNT1CDK9HASPIN
SCHEMBL21274452 0.74 LRRK2 (0.53) LRRK2CHUKDYRK1ACCNT1CDK9
SCHEMBL12120921 0.73 TYRO3 (0.42) HASPINRPS6KA5TYRO3DYRK1B
SCHEMBL18009669 0.73 RPS6KA5 (0.40) RPS6KA5TYRO3DYRK1B
SCHEMBL30475606 0.73 TYRO3 (0.42) HASPINRPS6KA5TYRO3DYRK1B
SCHEMBL14842412 0.73 AXL (0.47) CCNT1CDK9HASPINRPS6KA5TYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311896-A Pyrazolopyrimidine derivatives as kinase inhibitors 株式会社大熊制药 2019-02-05 CN disclosed