SCHEMBL2827688

SCHEMBL2827688

C[C@H](Cc1cccc(OCCC23CC4CC(CC(C4)C2)C3)c1)NC[C@H](O)c1ccc(O)c(C(N)=O)c1.NC(=O)c1cc([C@@H](O)CNCCc2cccc(OCCC34CC5CC(CC(C5)C3)C4)c2)ccc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 16/20 0.51
ADRB1 P08588 8/20 0.51
ADRA1D P25100 6/20 0.51
ADRA1A P35348 6/20 0.51
ADRA1B P35368 6/20 0.51
CYP2D6 P10635 2/20 0.51
ADRA2A P08913 2/20 0.51
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.51
HPGD P15428 2/20 0.51
HSD17B10 Q99714 2/20 0.51
DRD3 P35462 2/20 0.51
HTR1A P08908 1/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A4 P31645 1/20 0.51
OPRM1 P35372 1/20 0.51
HTR2B P41595 1/20 0.51
SLC6A3 Q01959 1/20 0.51
SIGMAR1 Q99720 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2748190 0.95 ADRB2 (0.53) ADRB2ADRB1ADRA1DADRA1AADRA1B
SCHEMBL2748515 0.93 ADRB2 (0.52) ADRB2ADRB1ADRA1DADRA1AADRA1B
SCHEMBL2827699 0.87 ADRB2 (0.63) ADRB2ADRB1ADRA1ACYP2D6DRD3
SCHEMBL2827697 0.87 ADRB2 (0.48) ADRB2ADRB1ADRA1ACYP2D6DRD3
SCHEMBL2747839 0.84 ADRB2 (0.43) ADRB2ADRB1ADRA1DADRA1AADRA1B
SCHEMBL2748296 0.84 ADRB2 (0.49) ADRB2ADRB1ADRA1DADRA1AADRA1B
SCHEMBL2748186 0.82 ADRB2 (0.57) ADRB2ADRB1ADRA1ACYP2D6HSD17B10
SCHEMBL2747898 0.82 ADRB2 (0.64) ADRB2ADRB1ADRB3
SCHEMBL2747476 0.82 ADRB2 (0.47) ADRB2ADRB1ADRB3
SCHEMBL2748512 0.79 ADRB2 (0.73) ADRB2ADRB1ADRA1ACYP2D6DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212276-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE BETA2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-08-04 EP disclosed
WO-2009068177-A1 DERIVATIVES OF 4-(2-AMINO-1 -HYDROXYETHYL)PHENOL AS AGONISTS OF THE β2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-06-04 WO disclosed