SCHEMBL28280658

SCHEMBL28280658

Cc1cc2nc(C=O)c(-c3ccccc3)nc2cc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.54
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 3/20 0.49
PDE10A Q9Y233 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PDGFRB P09619 1/20 0.46
KDR P35968 1/20 0.46
FLT3 P36888 1/20 0.46
NQO2 P16083 1/20 0.46
TDP1 Q9NUW8 2/20 0.43
TSHR P16473 1/20 0.43
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28278650 0.84 KDM4E (0.52) KDM4EALDH1A1PDE10AL3MBTL1NPC1
SCHEMBL30771455 0.82 KDM4E (0.68) ERBB2KDM4EALDH1A1PDE10AL3MBTL1
SCHEMBL28043991 0.82 KDM4E (0.68) ERBB2KDM4EALDH1A1PDE10AL3MBTL1
SCHEMBL28277283 0.80 NOS3 (0.44) ERBB2KDM4EALDH1A1L3MBTL1RAB9A
SCHEMBL12553478 0.80 ERBB2 (0.66) ERBB2KDM4EALDH1A1PDE10AL3MBTL1
SCHEMBL1302744 0.78 ERBB2 (0.64) ERBB2KDM4EALDH1A1PDE10AL3MBTL1
SCHEMBL6216319 0.77 ERBB2 (0.62) ERBB2KDM4EALDH1A1PDE10AL3MBTL1
SCHEMBL7935213 0.72 CYP3A4 (0.43) KDM4EALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL28281957 0.71 KDM4E (0.62) KDM4EALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL28278673 0.71 KDM4E (0.41) KDM4EALDH1A1L3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422699-A A kind of synthetic method of alpha-keto amide class compound 浙江工业大学 2019-03-05 CN disclosed