SCHEMBL28280894

SCHEMBL28280894

Clc1ccc(-c2cncnc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.56
KMT2A Q03164 2/20 0.49
MAPK10 P53779 2/20 0.49
MAPK9 P45984 1/20 0.49
USP2 O75604 1/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
CDC25B P30305 1/20 0.44
KCNH2 Q12809 1/20 0.41
MAPK14 Q16539 1/20 0.41
PTGS2 P35354 1/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TDO2 P48775 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4814511 0.83 NPSR1 (0.59) NPSR1KMT2AMAPK10MAPK9
SCHEMBL5215089 0.79 MAPK9 (0.56) KMT2AMAPK10MAPK9USP2CYP1A2
SCHEMBL30599018 0.79 MAPK9 (0.56) KMT2AMAPK10MAPK9USP2CYP1A2
SCHEMBL3311451 0.78 CYP1A2 (0.43) NPSR1KMT2AMAPK10USP2CYP1A2
SCHEMBL2424040 0.78 DGAT1 (0.62) NPSR1KMT2ACYP1A2KCNH2ALDH1A1
SCHEMBL10012834 0.78 NPSR1 (0.44) NPSR1KMT2AMAPK10USP2CYP1A2
SCHEMBL30782543 0.78 DGAT1 (0.62) NPSR1KMT2ACYP1A2KCNH2ALDH1A1
SCHEMBL3296530 0.78 NPSR1 (0.45) NPSR1KMT2AMAPK9USP2CYP1A2
SCHEMBL6323276 0.75 NPSR1 (0.51) NPSR1KMT2AMAPK10MAPK9KCNH2
SCHEMBL2275178 0.74 MAPK9 (0.51) NPSR1KMT2AMAPK10MAPK9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476599-A Guanidine derivatives and its medical usage 东丽株式会社 2019-03-15 CN disclosed