SCHEMBL2828124

SCHEMBL2828124

C[C@@H](Cc1ccc(OCC(F)(F)c2ccccc2)cc1)NC[C@@H](O)c1ccc(O)c(CO)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 14/20 0.54
ADRB1 P08588 6/20 0.49
ADRB3 P13945 5/20 0.49
ADRA1A P35348 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1B P35368 1/20 0.49
CYP2C9 P11712 1/20 0.49
SLC2A1 P11166 2/20 0.48
CASP3 P42574 1/20 0.48
CASP6 P55212 1/20 0.48
DRD2 P14416 2/20 0.47
PGR P06401 1/20 0.47
SLC6A4 P31645 1/20 0.47
PTGS2 P35354 1/20 0.47
SLC6A3 Q01959 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13232142 1.00 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL2828122 1.00 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL2795174 0.91 ADRB2 (0.59) ADRB2ADRB1ADRB3
SCHEMBL13170741 0.91 ADRB2 (0.59) ADRB2ADRB1ADRB3
SCHEMBL2795170 0.91 ADRB2 (0.59) ADRB2ADRB1ADRB3
SCHEMBL2853303 0.87 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL2853304 0.87 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL2853299 0.87 ADRB2 (0.54) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL2798250 0.87 ADRB3 (0.49) ADRB2ADRB1ADRB3ADRA1ACYP1A2
SCHEMBL4348119 0.87 ADRB3 (0.49) ADRB2ADRB1ADRB3ADRA1ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057122-B1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE 2 ADRENERGIC RECEPTOR ALMIRALL SA (ES) 2010-09-01 EP claimed