SCHEMBL28282010

SCHEMBL28282010

O=C(Nc1cc(Cl)c(F)cc1F)Oc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
KMT2A Q03164 4/20 0.54
MEN1 O00255 2/20 0.54
KDM4E B2RXH2 4/20 0.49
POLB P06746 1/20 0.49
ALDH1A1 P00352 5/20 0.46
HPGD P15428 2/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
ATM Q13315 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
MAOB P27338 1/20 0.46
CYP1A2 P05177 3/20 0.45
MAPT P10636 2/20 0.44
RAD51 Q06609 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22279199 0.88 NPC1 (0.62) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL29739633 0.87 NPC1 (0.52) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL27091711 0.87 NPC1 (0.52) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL5382561 0.85 NPC1 (0.52) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL24960688 0.85 NPC1 (0.52) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL29739599 0.84 NPSR1 (0.61) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL16907485 0.84 NPSR1 (0.61) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL9407126 0.83 NPSR1 (0.51) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL23635744 0.82 NPC1 (0.50) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL21319206 0.82 RAB9A (0.60) NPC1RAB9ANPSR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057739-A Diazepinone derivatives and their use in the treatment of hepatitis b infections 诺维拉治疗公司 2022-02-18 CN disclosed
CN-109641896-B Diazepinone derivatives and their use in the treatment of hepatitis b infections 诺维拉治疗公司 2021-09-21 CN disclosed
CN-109641896-A DIAZEPINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEPATITIS B INFECTIONS 诺维拉治疗公司 2019-04-16 CN disclosed