SCHEMBL28283271

SCHEMBL28283271

NC(=O)c1cnccc1NCCC(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT3 Q9NTG7 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
KDM4C Q9H3R0 10/20 0.43
KDM6B O15054 6/20 0.40
CD38 P28907 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.39
RPS6KB1 P23443 2/20 0.37
AURKA O14965 1/20 0.37
AURKB Q96GD4 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4A O75164 1/20 0.37
KDM4D Q6B0I6 1/20 0.37
TGFBR1 P36897 2/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15639467 0.85 SIRT3 (0.46) SIRT3TDP1KDM4CKDM6BCD38
SCHEMBL28283057 0.80 TP53 (0.43) KDM4CKDM6BKDM4EALDH1A1MAPT
SCHEMBL2122995 0.77 MKNK1 (0.57) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL3723389 0.77 SIRT3 (0.47) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL3716882 0.76 KDM4C (0.67) SIRT3TDP1KDM4CKDM6BRPS6KB1
SCHEMBL28284470 0.75 SIRT3 (0.49) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL22732130 0.75 SIRT3 (0.51) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL662028 0.74 SIRT3 (0.58) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL6757557 0.74 SIRT3 (0.58) SIRT3TDP1KDM4CKDM6BIRAK4
SCHEMBL7012861 0.74 RPS6KB1 (0.55) SIRT3TDP1KDM4CKDM6BRPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641906-A HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS 百时美施贵宝公司 2019-04-16 CN claimed
CN-106061967-B The nicotinamide compounds replaced through heteroaryl 百时美施贵宝公司 2019-04-19 CN disclosed
CN-109641906-A HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS 百时美施贵宝公司 2019-04-16 CN disclosed