SCHEMBL28286247

SCHEMBL28286247

CC(=O)Nc1ccc(NC(=O)O)cn1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.64
PTK2 Q05397 1/20 0.59
GAA P10253 2/20 0.53
CYP1A2 P05177 1/20 0.53
RAB9A P51151 8/20 0.50
SMN1; SMN2 Q16637 6/20 0.50
NPC1 O15118 5/20 0.50
MAPT P10636 3/20 0.49
HSD17B10 Q99714 1/20 0.48
KDM4E B2RXH2 1/20 0.48
NSD2 O96028 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
KIT P10721 1/20 0.46
KDR P35968 1/20 0.46
MAPK14 Q16539 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22501700 0.93 KMT2A (0.60) KMT2APTK2GAACYP1A2RAB9A
Hydrochloric Acid SCHEMBL28698696 0.91 KMT2A (0.58) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL13002752 0.84 PTK2 (0.61) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL14045205 0.82 RAB9A (0.72) KMT2ARAB9ASMN1; SMN2NPC1MAPT
SCHEMBL10222640 0.82 PTK2 (0.59) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL13698179 0.82 PTK2 (0.59) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL4516744 0.81 KMT2A (0.56) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL15223302 0.80 KMT2A (0.54) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL423961 0.79 RAB9A (0.75) KMT2APTK2GAACYP1A2RAB9A
SCHEMBL19766589 0.79 PTK2 (0.56) KMT2APTK2GAACYP1A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689664-B Tricyclic heteroaryl substituted quinoline and azaquinoline compounds as PAR4 inhibitors 百时美施贵宝公司 2022-04-15 CN claimed
CN-109689664-A The quinoline and azepine quinoline compound that tricyclic heteroaryl as PAR4 inhibitor replaces 百时美施贵宝公司 2019-04-26 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689664-B Tricyclic heteroaryl substituted quinoline and azaquinoline compounds as PAR4 inhibitors 百时美施贵宝公司 2022-04-15 CN disclosed
CN-109689664-A The quinoline and azepine quinoline compound that tricyclic heteroaryl as PAR4 inhibitor replaces 百时美施贵宝公司 2019-04-26 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed