SCHEMBL28287809

SCHEMBL28287809

Nc1ccc(C(=O)Nc2ccccc2)cc1N1CC[CH]CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 3/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC3 O15379 1/20 0.48
NCOR2 Q9Y618 1/20 0.48
PLAU P00749 2/20 0.47
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
PKM P14618 2/20 0.45
F2 P00734 1/20 0.45
PLG P00747 1/20 0.45
PLAT P00750 1/20 0.45
KLKB1 P03952 1/20 0.45
KLK1 P06870 1/20 0.45
PRSS1 P07477 1/20 0.45
NFKB1 P19838 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16146269 0.82 IRAK1 (0.60) HDAC2HDAC1HDAC3NCOR2PLAU
Hydrochloric Acid SCHEMBL16146311 0.81 IRAK1 (0.59) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL2949633 0.76 HDAC2 (0.63) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL29364540 0.76 HDAC2 (0.63) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL10280428 0.75 IRAK1 (0.45) HDAC2HDAC1HDAC3NCOR2ALDH1A1
SCHEMBL27498643 0.73 HDAC2 (0.59) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL9116112 0.72 HDAC2 (0.58) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL11701111 0.72 HDAC2 (0.58) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL9812753 0.71 HDAC2 (0.60) HDAC2HDAC1HDAC3NCOR2PLAU
SCHEMBL11200897 0.70 HDAC2 (0.59) HDAC2HDAC1HDAC3NCOR2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110003219-A Pyrazolo [1,5A] pyrimidine and thieno [3,2B] pyrimidine derivatives as IRAK4 regulator 弗·哈夫曼-拉罗切有限公司 2019-07-12 CN disclosed
CN-105367577-B Pyrazolo [1,5A] pyrimidine and thieno [3,2B] pyrimidine derivatives as IRAK4 regulator 弗·哈夫曼-拉罗切有限公司 2019-04-23 CN disclosed