SCHEMBL28290639

SCHEMBL28290639

O=Cc1cc(C(F)(C(F)(F)F)C(F)(F)F)ccc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
CYP3A4 P08684 2/20 0.41
ALOX15 P16050 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
PRKDC P78527 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ERN1 O75460 4/20 0.39
TDP1 Q9NUW8 2/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
TXNRD1 Q16881 1/20 0.38
TXNRD3 Q86VQ6 1/20 0.38
TXNRD2 Q9NNW7 1/20 0.38
ATM Q13315 1/20 0.36
ALDH5A1 P51649 1/20 0.36
ABAT P80404 1/20 0.36
VCAM1 P19320 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30849251 0.87 ALDH1A1 (0.47) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL17802484 0.87 ALDH1A1 (0.47) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL4596001 0.78 ERN1 (0.44) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL29910964 0.78 MAPT (0.50) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL6690245 0.78 MAPT (0.50) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL6452676 0.78 TDP1 (0.56) ALDH1A1CYP3A4ALOX15MAPTTDP1
SCHEMBL29404556 0.77 CYP3A4 (0.42) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL11126763 0.75 TDP1 (0.46) ALDH1A1CYP3A4ALOX15KDM4EMAPT
SCHEMBL19878494 0.75 ALDH1A1 (0.55) ALDH1A1CYP3A4ALOX15MAPTTDP1
SCHEMBL1094913 0.74 ALDH1A1 (0.41) ALDH1A1CYP3A4ALOX15KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808075-B Preparation method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-12-08 CN disclosed
CN-111704604-B Preparation method of pyridine quinazoline 湖南速博生物技术有限公司 2020-11-17 CN disclosed
CN-111808075-A Preparation method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-10-23 CN disclosed
CN-111533701-B Synthetic method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-10-16 CN disclosed
CN-111704604-A Preparation method of pyridine quinazoline 湖南速博生物技术有限公司 2020-09-25 CN disclosed
CN-111533701-A Synthetic method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-08-14 CN disclosed
CN-110698416-B Preparation method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-03-20 CN disclosed
CN-110698416-A Preparation method of pyridine quinazoline intermediate 湖南速博生物技术有限公司 2020-01-17 CN disclosed
CN-109705094-A A kind of preparation method of pyridine quinazoline 湖南速博生物技术有限公司 2019-05-03 CN disclosed