SCHEMBL28290672

SCHEMBL28290672

O=c1cc(N2CCC(c3nccs3)C2)c2ccncc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.40
CHEK1 O14757 3/20 0.37
CHEK2 O96017 3/20 0.37
PDE9A O76083 3/20 0.34
KDM4C Q9H3R0 1/20 0.34
CNR1 P21554 1/20 0.34
AOC3 Q16853 1/20 0.33
DRD4 P21917 2/20 0.32
PBK Q96KB5 1/20 0.32
SPR P35270 1/20 0.32
AOC2 O75106 1/20 0.32
PIK3C3 Q8NEB9 1/20 0.32
CYP17A1 P05093 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22298291 0.80 PDE9A (0.42) KDM5ACHEK1CHEK2PDE9AKDM4C
SCHEMBL22871692 0.78 PDE9A (0.60) KDM5APDE9A
SCHEMBL20870564 0.78 PDE9A (0.60) KDM5APDE9A
SCHEMBL23336509 0.78 PDE9A (0.60) KDM5APDE9A
SCHEMBL4751829 0.71 KDR (0.58) KDM5APDE9ADRD4
SCHEMBL28290751 0.71 KDM5A (0.44) KDM5ACHEK1CHEK2PDE9AKDM4C
SCHEMBL22225310 0.65 PDE9A (0.47) PDE9A
SCHEMBL17738664 0.64 PSEN1 (0.36) AOC3DRD4
SCHEMBL418629 0.64 KDM4E (0.47)
SCHEMBL24275785 0.63 PDE9A (0.44) PDE9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109575016-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-04-05 CN disclosed