SCHEMBL28290751

SCHEMBL28290751

CCOC1CCN(c2cc(=O)[nH]c3cnccc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 3/20 0.44
KDM5B Q9UGL1 1/20 0.38
CHEK1 O14757 2/20 0.38
CHEK2 O96017 2/20 0.38
BRD4 O60885 3/20 0.37
KDR P35968 1/20 0.36
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
CHUK O15111 1/20 0.36
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
PDE9A O76083 3/20 0.35
VNN1 O95497 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751829 0.78 KDR (0.58) KDM5AKDRADORA3CHUKPDE9A
SCHEMBL28290672 0.71 KDM5A (0.40) KDM5ACHEK1CHEK2PDE9AKDM4C
SCHEMBL4753880 0.68 KDR (0.61) KDM5ABRD4KDR
SCHEMBL19984551 0.67 KDM5A (0.67) KDM5AKDM5BADORA3ADORA2AADORA1
SCHEMBL30474111 0.67 KDM5A (0.67) KDM5AKDM5BADORA3ADORA2AADORA1
SCHEMBL20012152 0.64 GRIA1 (0.38) ADORA1PDE10A
SCHEMBL3242090 0.63 KDM5A (1.00) KDM5AKDM5BADORA3ADORA2AADORA1
SCHEMBL4756721 0.63 KDM5A (0.65) KDM5ACHUK
SCHEMBL30064094 0.63 KDM5A (1.00) KDM5AKDM5BADORA3ADORA2AADORA1
SCHEMBL246359 0.63 KDM5A (0.65) KDM5AKDM5BADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109575016-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-04-05 CN disclosed