SCHEMBL2829190

SCHEMBL2829190

CC(=O)c1cnc2c(Cl)cccc2c1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.55
NR1H2 P55055 12/20 0.52
NR1H3 Q13133 12/20 0.52
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
ALDH1A1 P00352 4/20 0.43
HTT P42858 3/20 0.43
HPGD P15428 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
DHODH Q02127 1/20 0.43
MAPT P10636 1/20 0.43
PPARG P37231 1/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2720744 0.85 HAVCR2 (0.50) HAVCR2NR1H2NR1H3ALDH1A1NPSR1
SCHEMBL2719758 0.82 CCNB2 (0.43) HAVCR2NR1H2NR1H3CCNB2CDK1
SCHEMBL2717720 0.81 HAVCR2 (0.57) HAVCR2NR1H2NR1H3CDK5SMN1; SMN2
SCHEMBL2729630 0.78 HAVCR2 (0.46) HAVCR2NR1H2NR1H3CDK5
SCHEMBL29611938 0.78 SMN1; SMN2 (0.66) NR1H2NR1H3CCNB2CDK1CCNB1
SCHEMBL2720220 0.78 SMN1; SMN2 (0.66) NR1H2NR1H3CCNB2CDK1CCNB1
SCHEMBL28623357 0.77 HAVCR2 (0.51) HAVCR2SMN1; SMN2MAPT
SCHEMBL1124612 0.76 NR1H2 (0.62) HAVCR2NR1H2NR1H3ALDH1A1HTT
SCHEMBL327460 0.75 NR1H2 (0.44) HAVCR2NR1H2NR1H3DHODHPPARG
SCHEMBL1125783 0.75 NR1H2 (0.75) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed