SCHEMBL28293431

SCHEMBL28293431

O=C(OCc1ccccc1)n1c(C2CO2)cc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.49
MAOA P21397 1/20 0.49
RCOR1 Q9UKL0 1/20 0.49
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
HTR2C P28335 1/20 0.42
CYP2C19 P33261 1/20 0.41
P2RX4 Q99571 2/20 0.41
P2RX1 P51575 1/20 0.41
P2RX3 P56373 1/20 0.41
CCR2 P41597 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PREP P48147 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3831363 0.78 KDM1A (0.56) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL7170567 0.78 KDM1A (0.48) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL28460969 0.76 KDM1A (0.47) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL10975824 0.76 POLB (0.43) MEN1KMT2ANPC1RAB9ACYP2C19
SCHEMBL8791569 0.73 KDM1A (0.52) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL19788743 0.72 P2RX4 (0.46) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL5241641 0.71 KDM1A (0.46) KDM1AMAOARCOR1MEN1KMT2A
SCHEMBL2530349 0.70 ALDH1A1 (0.50) MEN1KMT2ANPSR1SMN1; SMN2NPC1
SCHEMBL22675703 0.68 ALDH1A1 (0.55) MEN1KMT2ANPSR1SMN1; SMN2NPC1
SCHEMBL20628724 0.68 NR1H2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106674222-B A kind of chiral tricyclic ketone amine compound and its synthetic method and application 华东师范大学 2019-05-17 CN disclosed
CN-106674222-A Chiral tricyclic keto-amine compound as well as synthetic method and application thereof 华东师范大学 2017-05-17 CN disclosed