SCHEMBL28293604

SCHEMBL28293604

O=C(c1cccc(NS(=O)(=O)O)c1F)c1c[nH]c2ncccc12

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.52
CYP3A4 P08684 4/20 0.49
MAP2K1 Q02750 1/20 0.47
KDR P35968 1/20 0.47
BRAF P15056 2/20 0.46
NEK2 P51955 2/20 0.43
CNR2 P34972 1/20 0.40
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL297930 0.85 CYP2C9 (0.67) CYP2C9CYP3A4MAP2K1KDRBRAF
SCHEMBL28293606 0.84 BRAF (0.63) CYP2C9CYP3A4MAP2K1KDRBRAF
SCHEMBL30374918 0.84 CYP2C9 (0.56) CYP2C9CYP3A4MAP2K1KDRBRAF
SCHEMBL29652320 0.84 CYP2C9 (0.47) CYP2C9CYP3A4MAP2K1KDRBRAF
SCHEMBL15549990 0.83 MAP2K1 (0.48) CYP2C9CYP3A4MAP2K1KDRBRAF
SCHEMBL3509981 0.80 MAP2K1 (0.52) CYP2C9MAP2K1KDRBRAFNEK2
SCHEMBL3509976 0.80 MAP2K1 (0.52) CYP2C9MAP2K1KDRBRAFNEK2
SCHEMBL27708260 0.78 MAP2K1 (0.71) MAP2K1KDRBRAFNEK2CNR2
SCHEMBL288197 0.77 CYP2C9 (0.61) CYP2C9CYP3A4BRAF
SCHEMBL857351 0.76 MAP2K1 (0.57) CYP2C9MAP2K1KDRBRAFNEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109608450-A The synthesis of pyrrolo- [2,3-B] pyridine 普莱希科公司 2019-04-12 CN disclosed