SCHEMBL28294346

SCHEMBL28294346

CC(C)(O)CNC(=O)c1cc[c]cn1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.41
SCN9A Q15858 4/20 0.39
CFTR P13569 1/20 0.36
NAMPT P43490 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL749356 0.82 CNR1 (0.42)
SCHEMBL422451 0.76 CNR1 (0.38) SCN9A
SCHEMBL30975219 0.74 KMT2A (0.58)
SCHEMBL18279086 0.74 KMT2A (0.58)
SCHEMBL4772592 0.72 IL1B (0.36) SCN9A
SCHEMBL752887 0.72 CHRM2 (0.44)
SCHEMBL29085188 0.72 KDM4E (0.50) CNR2SCN9ACFTR
SCHEMBL30064984 0.72 KDM4E (0.50) CNR2SCN9ACFTR
SCHEMBL27720298 0.72 HIF1A (0.59)
SCHEMBL16277582 0.71 P4HTM (0.45) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed