SCHEMBL28295464

SCHEMBL28295464

CSCC[C@@H]1CNc2ccc(Cl)cc2C(c2ccccc2)=N1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 13/20 0.54
CCKBR P32239 2/20 0.47
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
ALB P02768 1/20 0.46
KMT2A Q03164 1/20 0.46
CNR1 P21554 1/20 0.46
NTSR1 P30989 1/20 0.46
OPRK1 P41145 1/20 0.46
PDE4D Q08499 1/20 0.46
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297191 1.00 CHRM1 (0.54) CHRM1CCKBRMEN1LMNAALB
SCHEMBL11684302 0.80 CHRM1 (0.62) CHRM1CCKBRMEN1LMNAALB
SCHEMBL28297259 0.80 CHRM1 (0.68) CHRM1CCKBRMEN1LMNAALB
SCHEMBL28297190 0.79 CHRM1 (0.64) CHRM1CCKBRMEN1LMNAALB
SCHEMBL21272215 0.79 CHRM1 (0.78) CHRM1CCKBRMEN1LMNAALB
SCHEMBL21272066 0.79 CHRM1 (0.78) CHRM1CCKBRMEN1LMNAALB
SCHEMBL21272106 0.78 CCKBR (0.70) CHRM1CCKBRMEN1LMNAALB
SCHEMBL11826012 0.78 CCKBR (0.70) CHRM1CCKBRMEN1LMNAALB
SCHEMBL21272237 0.78 CCKBR (0.70) CHRM1CCKBRMEN1LMNAALB
SCHEMBL7572862 0.77 MEN1 (0.52) CHRM1CCKBRMEN1LMNAALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN claimed
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed