SCHEMBL28295940

SCHEMBL28295940

NC(=O)CCc1ccc(-c2ccsc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.47
CYP17A1 P05093 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
FFAR1 O14842 1/20 0.43
CHEK1 O14757 1/20 0.43
CYP2E1 P05181 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2B6 P20813 1/20 0.41
CAPN1 P07384 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
KCNH2 Q12809 1/20 0.40
HDAC2 Q92769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696420 0.85 FFAR1 (0.62) CYP17A1CYP11B1CYP11B2FFAR1CYP2E1
SCHEMBL28295990 0.83 CA2 (0.50) CHEK2CYP17A1CYP11B1CYP11B2CYP2E1
SCHEMBL2102408 0.80 TAAR1 (0.55) CAPN1ALDH1A1LMNAHDAC6HDAC8
SCHEMBL27841461 0.80 FFAR1 (0.44) CHEK2CYP17A1CYP11B1CYP11B2FFAR1
Hydrochloric Acid SCHEMBL5347350 0.79 TAAR1 (0.53) CAPN1ALDH1A1LMNAHDAC6HDAC8
SCHEMBL5801662 0.77 FFAR1 (0.71) FFAR1LMNAHDAC1MMP2MMP9
SCHEMBL20399733 0.77 HDAC2 (0.62) FFAR1CAPN1ALDH1A1LMNAHDAC2
SCHEMBL4612023 0.77 CYP17A1 (0.53) CHEK2CYP17A1CYP11B1CYP11B2CYP2E1
SCHEMBL4591629 0.75 MAOB (0.55) FFAR1CAPN1ALDH1A1LMNAHDAC1
SCHEMBL27988046 0.75 MAOB (0.55) FFAR1CAPN1ALDH1A1LMNAHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776537-A Purinedione as WNT pathway modulators 新加坡科技研究局 2019-05-21 CN disclosed