SCHEMBL28296292

SCHEMBL28296292

N#Cc1ccnc(Cl)c1Br

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.40
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.34
KMO O15229 1/20 0.34
MEN1 O00255 1/20 0.34
CSNK1A1 P48729 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
SLC1A5 Q15758 1/20 0.33
GRM4 Q14833 1/20 0.32
CYP11B2 P19099 2/20 0.32
KHK P50053 1/20 0.32
TRPV4 Q9HBA0 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
CDC42BPA Q5VT25 1/20 0.31
CDC42BPB Q9Y5S2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL846091 0.78 LRRK2 (0.42) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL30007698 0.78 LRRK2 (0.42) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL1119092 0.75 FFAR1 (0.42) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL245839 0.75 CSNK1A1 (0.41) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL31321212 0.75 CSNK1A1 (0.41) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL30211311 0.75 LRRK2 (0.40) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL3287530 0.75 LRRK2 (0.40) LRRK2ALDH1A1NPSR1TDP1KMT2A
SCHEMBL27810450 0.71 BCL6 (0.37) LRRK2ALDH1A1TDP1KMT2AMEN1
SCHEMBL4475014 0.71 KDM4E (0.40) LRRK2ALDH1A1TDP1KMOCYP11B2
SCHEMBL25297122 0.71 KDM4E (0.33) LRRK2ALDH1A1NPSR1TDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843891-A Oxadiazolopyridine derivatives as ghrelin O-acyltransferase (GOAT) inhibitors 勃林格殷格翰国际有限公司 2019-06-04 CN disclosed