SCHEMBL2829763

SCHEMBL2829763

Cc1cc(C(C)(C)C)c2c(c1)C(O)(C(F)(F)F)C(=O)O2.Cc1ccc(O)c(C(C)(C)C)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.62
GABBR1 Q9UBS5 1/20 0.62
PDK2 Q15119 6/20 0.36
KDM4E B2RXH2 1/20 0.35
RAD52 P43351 1/20 0.35
ATM Q13315 1/20 0.35
ALDH1A1 P00352 3/20 0.35
TYR P14679 2/20 0.35
NR1I2 O75469 1/20 0.35
LMNA P02545 1/20 0.35
CYP2C9 P11712 1/20 0.35
MIF P14174 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
NFE2L2 Q16236 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HPGD P15428 2/20 0.34
CA2 P00918 1/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829152 0.90 GABBR2 (0.74) GABBR2GABBR1PDK2KDM4ERAD52
SCHEMBL2829154 0.90 GABBR2 (0.74) GABBR2GABBR1PDK2KDM4ERAD52
SCHEMBL2829157 0.90 GABBR2 (0.74) GABBR2GABBR1PDK2KDM4ERAD52
SCHEMBL2828609 0.83 GABBR2 (0.81) GABBR2GABBR1ALDH1A1TYRNR1I2
SCHEMBL2875028 0.81 GABBR2 (0.58) GABBR2GABBR1PDK2ATMALDH1A1
SCHEMBL2371842 0.77 GABBR2 (1.00) GABBR2GABBR1HSP90AA1
SCHEMBL2371847 0.77 GABBR2 (1.00) GABBR2GABBR1HSP90AA1
SCHEMBL2371840 0.77 GABBR2 (1.00) GABBR2GABBR1HSP90AA1
SCHEMBL30618192 0.77 GABBR2 (1.00) GABBR2GABBR1HSP90AA1
SCHEMBL2831256 0.74 GABBR2 (0.69) GABBR2GABBR1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1915357-B1 2-HYDROXY-PROPIONIC ACID DERIVATIVES AND 3-HYDROXY-BENZOFURAN-2-ONE DERIVATIVES WITH AFFINITY FOR THE GABA-B-RECEPTOR HOFFMANN LA ROCHE (CH) 2010-09-08 EP disclosed