SCHEMBL28297791

SCHEMBL28297791

Fc1ccc(-c2[nH]c3ncccc3c2F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.67
MAPK13 O15264 2/20 0.67
MAPK12 P53778 2/20 0.67
MAPK11 Q15759 2/20 0.67
MAPT P10636 3/20 0.44
GSK3B P49841 2/20 0.41
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
GSK3A P49840 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
AURKA O14965 1/20 0.41
PARP1 P09874 1/20 0.41
SERPINE1 P05121 1/20 0.41
HPGD P15428 1/20 0.40
BCHE P06276 1/20 0.40
CDC7 O00311 1/20 0.40
ROCK2 O75116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27546673 0.80 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11
SCHEMBL6250930 0.80 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11
SCHEMBL858101 0.74 MAPK14 (0.63) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL7921814 0.72 ADORA2A (0.76) MAPK14MAPK13MAPK12MAPK11GSK3B
SCHEMBL25029271 0.71 ALDH1A1 (0.54) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL1780573 0.70 MAPK13 (0.59) MAPK14MAPK13MAPK12MAPK11GSK3B
SCHEMBL1777550 0.70 MAPK13 (0.48) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL10395104 0.70 CDC7 (0.70) GSK3BCDK5CDK5R1CDC7ROCK2
SCHEMBL6525744 0.70 AURKA (0.60) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL6246075 0.69 MAPK14 (0.66) MAPK14MAPK13MAPK12MAPK11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106854205-B Inhibitors of influenza virus replication and methods of use and uses thereof 广东东阳光药业有限公司 2019-07-09 CN disclosed
CN-109748915-A Inhibitors of influenza viruses replication and its application method and purposes 广东东阳光药业有限公司 2019-05-14 CN disclosed