SCHEMBL28298506

SCHEMBL28298506

CC1(c2ccccc2)CCNC1.NC=S

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.49
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A3 Q01959 1/20 0.43
OPRM1 P35372 3/20 0.43
DRD2 P14416 1/20 0.37
HTR2C P28335 1/20 0.37
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
OPRL1 P41146 2/20 0.33
BACE1 P56817 1/20 0.33
TACR1 P25103 1/20 0.33
OPRK1 P41145 1/20 0.32
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331091 0.89 HTR2A (0.59) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL27225389 0.89 HTR2A (0.59) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL27099782 0.89 HTR2A (0.59) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL3438951 0.79 HTR2A (0.50) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL19122010 0.79 HTR2A (0.50) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL737635 0.78 OPRM1 (0.61) HTR2ACYP2D6OPRM1OPRL1TACR1
Hydrochloric Acid SCHEMBL8587704 0.77 HTR2A (0.48) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
Hydrochloric Acid SCHEMBL10007993 0.76 OPRM1 (0.59) HTR2ACYP2D6OPRM1OPRL1TACR1
SCHEMBL19074637 0.75 SLC6A2 (0.51) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3
Hydrochloric Acid SCHEMBL5874274 0.74 CYP2D6 (0.46) HTR2ASLC6A2SLC6A4CYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed