SCHEMBL28301987

SCHEMBL28301987

Nc1nc(N)c2ncn(C3CCNC3)c2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHCY P23526 3/20 0.46
ADORA2A P29274 5/20 0.46
PI4KA P42356 3/20 0.43
PI4K2B Q8TCG2 3/20 0.43
PI4K2A Q9BTU6 3/20 0.43
PI4KB Q9UBF8 3/20 0.43
ADORA3 P0DMS8 3/20 0.43
ADORA1 P30542 3/20 0.43
ADORA2B P29275 2/20 0.43
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNE1 P24864 2/20 0.42
CDK2 P24941 2/20 0.42
SRC P12931 3/20 0.42
EGFR P00533 2/20 0.42
ABL1 P00519 1/20 0.42
ABL2 P42684 1/20 0.42
DNMT1 P26358 1/20 0.41
HSP90B1 P14625 1/20 0.40
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29444625 0.92 ADORA2A (0.48) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL15941621 0.84 ADORA2A (0.63) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL15720194 0.82 ADORA2A (0.70) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL17352601 0.81 ADORA2A (0.65) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL2954550 0.80 ADORA2A (0.66) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL2952924 0.77 ADORA2A (0.51) AHCYADORA2API4KAPI4K2BPI4K2A
SCHEMBL2949862 0.77 ADORA2A (0.51) AHCYADORA2API4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL5626685 0.74 AHCY (0.48) AHCYADORA2API4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL7846299 0.74 AHCY (0.54) AHCYADORA2API4KAPI4K2BPI4K2A
Sulfuric Acid SCHEMBL9424495 0.74 CYP1A2 (0.63) AHCYADORA2API4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114149432-A Dual CLK/CDK1 inhibitors for cancer treatment 斯坦福国际研究院 2022-03-08 CN disclosed
CN-109937039-A DUAL CLK/CDK1 INHIBITORS FOR CANCER TREATMENT 斯坦福国际研究院 2019-06-25 CN disclosed