SCHEMBL28305545

SCHEMBL28305545

O=C1C(C=Cc2ccc(N(c3ccccc3)c3ccccc3)cc2)C(=O)N(c2ccccc2)C(=O)N1c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.39
KMT2A Q03164 8/20 0.39
ALDH1A1 P00352 7/20 0.39
MEN1 O00255 7/20 0.39
PKM P14618 4/20 0.39
NPSR1 Q6W5P4 4/20 0.39
APP P05067 4/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
MAPK1 P28482 3/20 0.39
PSMD14 O00487 2/20 0.39
THRB P10828 2/20 0.39
SNCA P37840 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MMP2 P08253 1/20 0.39
PPARG P37231 1/20 0.39
NCOA2 Q15596 1/20 0.39
NPC1 O15118 1/20 0.39
ALPG P10696 1/20 0.39
RECQL P46063 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28306761 0.82 APP (0.39) MAPTKMT2AALDH1A1MEN1PKM
SCHEMBL28306750 0.75 MAPT (0.44) MAPTKMT2AALDH1A1MEN1PKM
SCHEMBL806444 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL21922852 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL275803 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL101911 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL275802 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL14018370 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL14526617 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1
SCHEMBL13927945 0.69 RELA (0.60) MAPTKMT2AALDH1A1MEN1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110028456-B Barbituric acid derivative and preparation method and application thereof 齐鲁工业大学 2021-02-23 CN disclosed
CN-110028456-A A kind of barbituric acid derivatives and preparation method and application 齐鲁工业大学 2019-07-19 CN disclosed