SCHEMBL28308017

SCHEMBL28308017

CCCCCc1nc2cccc(Br)c2c(=O)[nH]1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.57
GPR84 Q9NQS5 5/20 0.43
POLB P06746 1/20 0.42
PARP2 Q9UGN5 2/20 0.42
TNKS2 Q9H2K2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28279923 0.84 TNKS2 (0.58) PARP1TNKS2
SCHEMBL28308034 0.84 PARP1 (0.57) PARP1GPR84PARP2TNKS2
SCHEMBL28307043 0.84 PARP1 (0.57) PARP1GPR84POLBPARP2TNKS2
SCHEMBL27764706 0.84 PARP1 (0.57) PARP1GPR84
SCHEMBL1586541 0.77 PARP1 (0.91) PARP1PARP2TNKS2
SCHEMBL30176861 0.76 PARP1 (0.89) PARP1PARP2TNKS2
SCHEMBL14621928 0.76 PARP1 (0.89) PARP1PARP2TNKS2
SCHEMBL22857122 0.76 PARP1 (0.89) PARP1PARP2TNKS2
SCHEMBL30176973 0.76 PARP1 (0.89) PARP1PARP2TNKS2
SCHEMBL28598382 0.76 PARP1 (0.89) PARP1PARP2TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041306-A 4- hydroxyl -2- quinolone-nitrogen-(4- quinazolinone) -3- carboxamides derivatives 中国医学科学院药物研究所 2019-07-23 CN disclosed