SCHEMBL28308019

SCHEMBL28308019

CCCc1nc2ccccc2c(=O)n1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.81
ATM Q13315 1/20 0.81
LMNA P02545 3/20 0.79
TSHR P16473 1/20 0.79
NPC1 O15118 4/20 0.61
KDM4E B2RXH2 2/20 0.59
RAB9A P51151 5/20 0.58
USP2 O75604 2/20 0.58
KMT2A Q03164 3/20 0.56
MEN1 O00255 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
MAPT P10636 2/20 0.56
HTT P42858 2/20 0.56
ALDH1A1 P00352 1/20 0.56
GAA P10253 1/20 0.54
GLA P06280 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5928664 0.91 SMN1; SMN2 (0.92) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL28308015 0.90 SMN1; SMN2 (1.00) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL28307048 0.88 LMNA (1.00) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL28308021 0.88 LMNA (1.00) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL3714715 0.87 SMN1; SMN2 (0.71) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL14743414 0.86 SMN1; SMN2 (0.69) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL18017411 0.83 HDAC6 (0.71) SMN1; SMN2ATMLMNATSHRKDM4E
SCHEMBL5928772 0.81 NPC1 (0.64) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL28677827 0.80 SMN1; SMN2 (0.62) SMN1; SMN2ATMLMNATSHRNPC1
SCHEMBL5928915 0.80 NPC1 (0.72) SMN1; SMN2ATMLMNATSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041306-B 4-hydroxy-2-quinolone-N- (4-quinazolinone) -3-carboxamide derivatives 中国医学科学院药物研究所 2022-01-11 CN disclosed
CN-110041306-A 4- hydroxyl -2- quinolone-nitrogen-(4- quinazolinone) -3- carboxamides derivatives 中国医学科学院药物研究所 2019-07-23 CN disclosed