Pyrazole

Pyrazole

SCHEMBL28308907

O=CNc1nccs1.c1cn[nH]c1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 8/20 0.36
LMNA P02545 2/20 0.36
TSHR P16473 1/20 0.36
NPC1 O15118 7/20 0.36
SMN1; SMN2 Q16637 6/20 0.35
GAA P10253 1/20 0.35
ACP1 P24666 1/20 0.35
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
AURKA O14965 1/20 0.35
PIM1 P11309 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
KDM4E B2RXH2 2/20 0.35
TP53 P04637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL970110 0.83
Bromide SCHEMBL28645412 0.81
Glyoxylate SCHEMBL8429578 0.73 HTT (0.51) ALDH1A1MAPTKMT2AMEN1RAB9A
Acetic Acid SCHEMBL8425256 0.73 HTT (0.55) ALDH1A1MAPTKMT2AMEN1RAB9A
Aminothiazole SCHEMBL28835087 0.71 ALDH1A1 (0.60) ALDH1A1TSHR
Formanilide SCHEMBL28303566 0.70 ALDH1A1 (0.61) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL28855042 0.69
Pyrazole SCHEMBL29006140 0.68
Pyrazole SCHEMBL27834927 0.68
Pyrazole SCHEMBL27757216 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906226-A Heterocyclic compounds and their use in the prevention or treatment of bacterial infections 拜欧蒂姆公司 2019-06-18 CN disclosed