SCHEMBL28309779

SCHEMBL28309779

OCC(O)Cc1cccc2ncccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
MAPT P10636 1/20 0.44
CYP19A1 P11511 1/20 0.42
TBXAS1 P24557 1/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
POLB P06746 1/20 0.39
NSD2 O96028 1/20 0.38
SCN9A Q15858 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
GLS O94925 1/20 0.37
CYP3A4 P08684 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28308989 0.81 KDM4E (0.45) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL3136413 0.80 KDM4E (0.56) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL12749711 0.77 KDM4E (0.48) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL5495469 0.75 CYP19A1 (0.54) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL3817705 0.74 MAPT (0.54) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL23844520 0.74 KDM4E (0.41) KDM4EMAPTCYP19A1TBXAS1ALDH1A1
SCHEMBL5583861 0.74 KDM4E (0.42) KDM4EMAPTALDH1A1LMNAHTT
SCHEMBL14456318 0.74 KDM4E (0.38) KDM4EMAPTMEN1KMT2ASCN9A
SCHEMBL14656677 0.74 CYP1A2 (0.42) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL9183907 0.73 LOXL2 (0.61) KDM4EMAPTALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814040-B The condensed 1,4- dihydro two of inhibitor as thermal excited transcryption factor 1 dislikes ene derivative 癌症研究科技有限公司 2019-07-30 CN disclosed