SCHEMBL28326883

SCHEMBL28326883

COc1ccc(-c2cncc3ccccc23)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.68
CYP11B2 P19099 7/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2B6 P20813 1/20 0.68
CYP2C19 P33261 1/20 0.68
TLR9 Q9NR96 1/20 0.61
ERN1 O75460 1/20 0.60
PRKCZ Q05513 1/20 0.54
ACACA Q13085 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
CYP17A1 P05093 4/20 0.50
PRKCQ Q04759 1/20 0.49
ADORA1 P30542 1/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821959 0.85 CYP1A2 (0.54) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL10591476 0.81 FLT3 (0.54) ACACAMEN1KMT2AKDM4EALDH1A1
SCHEMBL4214556 0.80 CYP11B1 (0.78) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL29501832 0.80 CYP11B1 (0.78) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8503236 0.78 CYP11B1 (0.76) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL22575717 0.78 TLR9 (1.00) TLR9
SCHEMBL2203843 0.78 CYP17A1 (0.58) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL29501876 0.77 CYP11B1 (0.74) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL7299965 0.76 CYP11B1 (0.67) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6
SCHEMBL12767004 0.75 ERN1 (1.00) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073744-B Novel heterocyclic compounds as bromine structural domain inhibitor ZENITH EPIGENETICS CORP. (CA) 2019-11-08 CN disclosed