SCHEMBL7299965

SCHEMBL7299965

COc1ccc2cc(-c3cncc4ccccc34)ccc2n1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 13/20 0.67
CYP11B2 P19099 13/20 0.67
CYP2D6 P10635 2/20 0.67
CYP2C9 P11712 2/20 0.67
CYP2B6 P20813 2/20 0.67
CYP2C19 P33261 2/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
ERN1 O75460 2/20 0.48
PRKCZ Q05513 1/20 0.48
ADORA1 P30542 1/20 0.47
CYP17A1 P05093 1/20 0.46
TLR9 Q9NR96 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
WNT1 P04628 1/20 0.41
DYRK1A Q13627 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501876 0.78 CYP11B1 (0.74) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL28326883 0.76 CYP11B1 (0.68) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL12695592 0.75 BACE1 (0.57) CYP11B1CYP11B2ADORA1CYP17A1MEN1
SCHEMBL31149547 0.75 ADORA1 (0.41) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL29501832 0.74 CYP11B1 (0.78) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL4214556 0.74 CYP11B1 (0.78) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
Hydrochloric Acid SCHEMBL8503236 0.73 CYP11B1 (0.76) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL21215634 0.73 CYP11B1 (0.52) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6
SCHEMBL7264558 0.72 CYP11B2 (0.64) CYP11B1CYP11B2CYP17A1DYRK1A
SCHEMBL5425408 0.72 CYP11B1 (0.65) CYP11B1CYP11B2CYP2D6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4898872-A Imidazo[4,5-b]pyridyl quinolone cardiac stimulants PFIZER INC. (US) 1990-02-06 US disclosed
EP-0290153-A1 Heterobicyclic quinolone derivatives Pfizer Limited (GB) 1988-11-09 EP disclosed