SCHEMBL28331817

SCHEMBL28331817

CCOc1c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c2c1F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 6/20 0.60
TOP2B Q02880 6/20 0.60
KCNH2 Q12809 5/20 0.56
GSK3B P49841 2/20 0.53
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
HPGD P15428 2/20 0.52
HSD17B10 Q99714 2/20 0.52
POLB P06746 2/20 0.52
OPRM1 P35372 2/20 0.52
PRKD3 O94806 1/20 0.52
ALOX15 P16050 1/20 0.52
CLK2 P49760 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
ADRB2 P07550 1/20 0.51
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328397 0.91 TOP2A (0.57) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL9263643 0.91 TOP2A (0.49) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL28408530 0.89 KCNH2 (0.61) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL6645463 0.83 TOP2A (0.60) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL500719 0.82 TOP2A (0.71) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL29463823 0.82 TOP2A (0.71) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL30804388 0.82 KDM4E (0.55) ALDH1A1KDM4EHPGDHSD17B10POLB
SCHEMBL29161420 0.82 KDM4E (0.55) ALDH1A1KDM4EHPGDHSD17B10POLB
SCHEMBL9383693 0.82 TOP2A (0.69) TOP2ATOP2BKCNH2GSK3BALDH1A1
SCHEMBL10330765 0.82 TOP2A (0.69) TOP2ATOP2BKCNH2GSK3BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110551124-B Quinolone compound or agriculturally and pharmaceutically acceptable salt thereof, and preparation method and application thereof 山东省联合农药工业有限公司 2021-01-08 CN disclosed
CN-110551124-A quinolone compound or agriculturally and pharmaceutically acceptable salt thereof, and preparation method and application thereof SHANDONG UNITED PESTICIDE IND CO LTD 2019-12-10 CN disclosed