SCHEMBL28332018

SCHEMBL28332018

COc1ccc(N(C(C)=O)c2ccc(OC)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.55
MEN1 O00255 1/20 0.54
TSHR P16473 1/20 0.54
KMT2A Q03164 1/20 0.54
ALDH1A1 P00352 1/20 0.50
HTT P42858 1/20 0.50
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
MAPT P10636 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
TP53 P04637 1/20 0.49
ESR2 Q92731 1/20 0.49
NOX1 Q9Y5S8 1/20 0.49
CA1 P00915 6/20 0.48
CA2 P00918 6/20 0.48
CA12 O43570 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31393785 0.92 KMT2A (0.66) POLBMEN1TSHRKMT2AALDH1A1
SCHEMBL10160616 0.88 KMT2A (0.60) POLBMEN1TSHRKMT2ACES2
SCHEMBL12037062 0.88 KMT2A (0.56) POLBMEN1TSHRKMT2AALDH1A1
SCHEMBL28904603 0.83 CA1 (0.48) POLBMEN1TSHRKMT2AALDH1A1
SCHEMBL2113106 0.83 CES2 (0.47) POLBMEN1TSHRKMT2AALDH1A1
SCHEMBL8057301 0.83 CES2 (0.50) POLBALDH1A1HTTCES2CES1
SCHEMBL4601283 0.83 CA1 (0.54) MEN1TSHRKMT2ACES2CES1
SCHEMBL3278204 0.81 KDM4E (0.56) POLBALDH1A1HTTCES2CES1
SCHEMBL3470955 0.81 CA1 (0.55) CES2CES1MAPTNPC1RAB9A
SCHEMBL11540415 0.81 CES2 (0.48) POLBTSHRALDH1A1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110382458-A Enamine compound and application thereof 国立研究开发法人科学技术振兴机构 2019-10-25 CN disclosed